TIDGN: A Transfer Learning Framework for Predicting Interactions of Intrinsically Disordered Proteins with High Conformational Dynamics.

Journal: Journal of chemical information and modeling
Published Date:

Abstract

Interactions between intrinsically disordered proteins (IDPs) are crucial for biological processes, such as intracellular liquid-liquid phase separation (LLPS). Experiments (e.g., NMR) and simulations used to study IDP interactions encounter a variety of difficulties, highlighting the necessity to develop relevant machine learning methods. However, reliable machine learning methods face the challenge resulting from the scarcity of available training data. In this work, we propose a transfer learning-based invariant geometric dynamic graph model, named TIDGN, for predicting IDP interactions. The model consists of a pretraining task module and a downstream task module. The pretraining task module learns the dynamic structural encoding of IDP monomers, which is then used by the downstream task module for interaction site prediction. The IDP monomer structure data set and the IDP interaction event data set are constructed using all-atom molecular dynamics (MD) simulations. The transfer learning strategy effectively enhances the model's performance. Both homotypic interactions and heterotypic interactions between two IDPs are considered in this work. Interestingly, TIDGN performs well for the heterotypic interaction prediction. Additionally, the feature ablation analysis emphasizes the importance of invariant geometric graph features. Taken together, our work demonstrates that the integration of transfer learning and the invariant geometric graph network offers a promising approach for addressing data scarcity challenges of IDP interaction prediction.

Authors

  • Jing Xiao
    Xiyuan Hospital, China Academy of Chinese Medical Sciences(CACMS), Beijing, China.
  • Guorong Hu
    School of Physics, Zhejiang University, Hangzhou 310058, P. R. China.
  • Xiaozhou Zhou
    Department of Urology, Urology Institute of PLA, Southwest Hospital, Third Military Medical University, Chongqing, China.
  • Yuchuan Zheng
    School of Physics, Zhejiang University, Hangzhou 310058, P. R. China.
  • Jingyuan Li
    Zhejiang Province Key Laboratory of Quantum Technology and Device, Institute of Quantitative Biology, Department of Physics, Zhejiang University, Hangzhou 310027, Zhejiang, China.