The isolation, bioactivity, and synthesis of natural products from with anti-HIV activities.

Journal: Frontiers in pharmacology
Published Date:

Abstract

Natural products isolated from have attracted considerable attention from the chemical community due to their unique structures and promising anti-HIV activities. Recent progresses in the isolation and bioactivity studies for these natural molecules were summarized comprehensively. From the 23 previously uncharacterized compounds isolated from the plant , litseaverticillol B demonstrated the most potent anti-HIV activity , with IC ranging from 2 to 3 μg/mL. Meanwhile, litseaverticillol E displayed the highest selectivity index (SI = 3.1), indicating a favorable balance between antiviral potency and cellular toxicity. The plausible biosynthetic pathways and the total synthetic approaches for the representative members (litseaverticillols) were introduced in detail.

Authors

  • Jia-Lei Yan
    School of Pharmacy and Food Engineering, Wuyi University, Jiangmen, China.
  • Huiru Nan
    School of Pharmacy and Food Engineering, Wuyi University, Jiangmen, China.
  • Xiaoyu Fang
    School of Pharmacy and Food Engineering, Wuyi University, Jiangmen, China.
  • Xiong-En Long
    School of Pharmacy and Food Engineering, Wuyi University, Jiangmen, China.
  • Yu Jiang
    School of Pharmacy and Food Engineering, Wuyi University, Jiangmen, China.
  • Junyang Liu
    School of Pharmacy and Food Engineering, Wuyi University, Jiangmen, China.

Keywords

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