Classification of alkaloids according to the starting substances of their biosynthetic pathways using graph convolutional neural networks.

Journal: BMC bioinformatics
Published Date:

Abstract

BACKGROUND: Alkaloids, a class of organic compounds that contain nitrogen bases, are mainly synthesized as secondary metabolites in plants and fungi, and they have a wide range of bioactivities. Although there are thousands of compounds in this class, few of their biosynthesis pathways are fully identified. In this study, we constructed a model to predict their precursors based on a novel kind of neural network called the molecular graph convolutional neural network. Molecular similarity is a crucial metric in the analysis of qualitative structure-activity relationships. However, it is sometimes difficult for current fingerprint representations to emphasize specific features for the target problems efficiently. It is advantageous to allow the model to select the appropriate features according to data-driven decisions for extracting more useful information, which influences a classification or regression problem substantially.

Authors

  • Ryohei Eguchi
    Division of Science and Technology, Graduate School of Science and Technology, Nara Institute of Science and Technology, Ikoma, Nara, 630-0192, Japan.
  • Naoaki Ono
    Data Science Center, Nara Institute of Science and Technology, Ikoma, Japan. nono@is.naist.jp.
  • Aki Hirai Morita
    Division of Science and Technology, Graduate School of Science and Technology, Nara Institute of Science and Technology, Ikoma, Nara, 630-0192, Japan.
  • Tetsuo Katsuragi
    Department of Computer Science and Engineering, Toyohashi University of Technology, Hibarigaoka, Tempaku-cho, Toyohashi, Aichi, 441-8580, Japan.
  • Satoshi Nakamura
    Radiation Safety and Quality Assurance Division, National Cancer Center Hospital, 5-1-1 Tsukiji, Chuo-ku, Tokyo, Japan.
  • Ming Huang
    College of Food Science and Technology, Nanjing Agricultural University, Nanjing 210095, China.
  • Md Altaf-Ul-Amin
    Graduate School of Science and Technology, Nara Institute of Science and Technology, Ikoma, Japan.
  • Shigehiko Kanaya
    Graduate School of Science and Technology, Nara Institute of Science and Technology, Ikoma, Japan.