Simplified and enhanced VCD analysis of cyclic peptides guided by artificial intelligence.

Journal: Physical chemistry chemical physics : PCCP
Published Date:

Abstract

Cyclic peptides are privileged structures in medicinal chemistry; however, their solution-state structure characterization is difficult. Vibrational circular dichroism (VCD) spectroscopy is a powerful alternative to NMR, but requires challenging calculations. We present a VCD approach guided by a genetic algorithm, which is simple, more effective, and has a higher conformer resolution.

Authors

  • João M Batista
    Federal University of São Paulo, Institute of Science and Technology, R. Talim 330, 12231-280, São José dos Campos-SP, Brazil. batista.junior@unifesp.br.
  • Valentin Paul Nicu
    ProVitam Foundation, Caisului Street 16, Cluj-Napoca, Romania. vp.nicu@gmail.com.