Fast and accurate prediction of partial charges using Atom-Path-Descriptor-based machine learning.

Journal: Bioinformatics (Oxford, England)
PMID:

Abstract

MOTIVATION: Partial atomic charges are usually used to calculate the electrostatic component of energy in many molecular modeling applications, such as molecular docking, molecular dynamics simulations, free energy calculations and so forth. High-level quantum mechanics calculations may provide the most accurate way to estimate the partial charges for small molecules, but they are too time-consuming to be used to process a large number of molecules for high throughput virtual screening.

Authors

  • Jike Wang
    School of Computer Science, Wuhan University, Wuhan, Hubei 430072, China.
  • Dongsheng Cao
    School of Pharmaceutical Sciences, Central South University, Changsha, China. oriental-cds@163.com.
  • Cunchen Tang
    School of Computer Science, Wuhan University, Wuhan, Hubei 430072, China.
  • Xi Chen
    Department of Critical care medicine, Shenzhen Hospital, Southern Medical University, Guangdong, Shenzhen, China.
  • Huiyong Sun
    College of Pharmaceutical Sciences, Zhejiang University , Hangzhou, Zhejiang 310058, China.
  • Tingjun Hou
    College of Pharmaceutical Sciences, Zhejiang University , Hangzhou, Zhejiang 310058, China.