AIMC Topic: Drug Discovery

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Prediction of hot spots towards drug discovery by protein sequence embedding with 1D convolutional neural network.

PloS one
Protein hotspot residues are key sites that mediate protein-protein interactions. Accurate identification of these residues is essential for understanding the mechanism from protein to function and for designing drug targets. Current research has mos...

Transforming drug discovery with a high-throughput AI-powered platform: A 5-year experience with Patrimony.

Drug discovery today
High-throughput computational platforms are being established to accelerate drug discovery. Servier launched the Patrimony platform to harness computational sciences and artificial intelligence (AI) to integrate massive multimodal data from internal ...

Artificial intelligence revolutionizing drug development: Exploring opportunities and challenges.

Drug development research
By harnessing artificial intelligence (AI) algorithms and machine learning techniques, the entire drug discovery process stands to undergo a profound transformation, offering a myriad of advantages. Foremost among these is the ability of AI to conduc...

First fully-automated AI/ML virtual screening cascade implemented at a drug discovery centre in Africa.

Nature communications
Streamlined data-driven drug discovery remains challenging, especially in resource-limited settings. We present ZairaChem, an artificial intelligence (AI)- and machine learning (ML)-based tool for quantitative structure-activity/property relationship...

Artificial intelligence for natural product drug discovery.

Nature reviews. Drug discovery
Developments in computational omics technologies have provided new means to access the hidden diversity of natural products, unearthing new potential for drug discovery. In parallel, artificial intelligence approaches such as machine learning have le...

An improved multi-modal representation-learning model based on fusion networks for property prediction in drug discovery.

Computers in biology and medicine
Accurate characterization of molecular representations plays an important role in the property prediction based on deep learning (DL) for drug discovery. However, most previous researches considered only one type of molecular representations, resulti...

A large-scale evaluation of NLP-derived chemical-gene/protein relationships from the scientific literature: Implications for knowledge graph construction.

PloS one
One area of active research is the use of natural language processing (NLP) to mine biomedical texts for sets of triples (subject-predicate-object) for knowledge graph (KG) construction. While statistical methods to mine co-occurrences of entities wi...

In silico co-crystal design: Assessment of the latest advances.

Drug discovery today
Pharmaceutical co-crystals represent a growing class of crystal forms in the context of pharmaceutical science. They are attractive to pharmaceutical scientists because they significantly expand the number of crystal forms that exist for an active ph...

Making the Case for Quantum Mechanics in Predictive Toxicology─Nearly 100 Years Too Late?

Chemical research in toxicology
The use of quantum mechanics (QM) has long been the norm to study covalent-binding phenomena in chemistry and biochemistry. The pharmaceutical industry leverages QM models explicitly in covalent drug discovery and implicitly to characterize short-ran...

DeepTPpred: A Deep Learning Approach With Matrix Factorization for Predicting Therapeutic Peptides by Integrating Length Information.

IEEE journal of biomedical and health informatics
The abuse of traditional antibiotics has led to increased resistance of bacteria and viruses. Efficient therapeutic peptide prediction is critical for peptide drug discovery. However, most of the existing methods only make effective predictions for o...