AI Medical Compendium Journal:
Current topics in medicinal chemistry

Showing 11 to 20 of 38 articles

Artificial Intelligence in Drug Design: Are We Still There?

Current topics in medicinal chemistry
BACKGROUND: The artificial intelligence (AI)-assisted design of drug candidates with novel structures and desired properties has received significant attention in the recent past, so related areas of forward prediction that aim to discover chemical m...

Artificial Intelligence Approaches in Drug Discovery: Towards the Laboratory of the Future.

Current topics in medicinal chemistry
The role of computational tools in the drug discovery and development process is becoming central, thanks to the possibility to analyze large amounts of data. The high throughput and affordability of current omics technologies, allowing quantitative ...

Computational Approaches for Investigating Disease-causing Mutations in Membrane Proteins: Database Development, Analysis and Prediction.

Current topics in medicinal chemistry
Membrane proteins (MPs) play an essential role in a broad range of cellular functions, serving as transporters, enzymes, receptors, and communicators, and about ~60% of membrane proteins are primarily used as drug targets. These proteins adopt either...

Machine Learning and Artificial Intelligence: A Paradigm Shift in Big Data-Driven Drug Design and Discovery.

Current topics in medicinal chemistry
BACKGROUND: The lengthy and expensive process of developing a novel medicine often takes many years and entails a significant financial burden due to its poor success rate. Furthermore, the processing and analysis of quickly expanding massive data ne...

Artificial Intelligence and Cheminformatics-Guided Modern Privileged Scaffold Research.

Current topics in medicinal chemistry
With the rapid development of computer science in scopes of theory, software, and hardware, artificial intelligence (mainly in form of machine learning and more complex deep learning) combined with advanced cheminformatics is playing an increasingly ...

Predicting Metabolic Reaction Networks with Perturbation-Theory Machine Learning (PTML) Models.

Current topics in medicinal chemistry
BACKGROUND: Checking the connectivity (structure) of complex Metabolic Reaction Networks (MRNs) models proposed for new microorganisms with promising properties is an important goal for chemical biology.

The Role of Machine Learning in Centralized Authorization Process of Nanomedicines in European Union.

Current topics in medicinal chemistry
BACKGROUND: Machine Learning (ML) has experienced an increasing use, given the possibilities to expand the scientific knowledge of different disciplines, such as nanotechnology. This has allowed the creation of Cheminformatic models capable of predic...

Machine Learning and Perturbation Theory Machine Learning (PTML) in Medicinal Chemistry, Biotechnology, and Nanotechnology.

Current topics in medicinal chemistry
Recently, different authors have reported Perturbation Theory (PT) methods combined with machine learning (ML) to obtain PTML (PT + ML) models. They have applied PTML models to the study of different biological systems. Here we present one state-of-a...

PTML Multi-Label Algorithms: Models, Software, and Applications.

Current topics in medicinal chemistry
By combining Machine Learning (ML) methods with Perturbation Theory (PT), it is possible to develop predictive models for a variety of response targets. Such combination often known as Perturbation Theory Machine Learning (PTML) modeling comprises a ...