An AI-assisted fluorescence microscopic system for screening mitophagy inducers by simultaneous analysis of mitophagic intermediates.

Journal: Nature communications
Published Date:

Abstract

Mitophagy, the selective autophagic elimination of mitochondria, is essential for maintaining mitochondrial quality and cell homeostasis. Impairment of mitophagy flux, a process involving multiple sequential intermediates, is implicated in the onset of numerous neurodegenerative diseases. Screening mitophagy inducers, particularly understanding their impact on mitophagic intermediates, is crucial for neurodegenerative disease treatment. However, existing techniques do not allow simultaneous visualization of distinct mitophagic intermediates in live cells. Here, we introduce an artificial intelligence-assisted fluorescence microscopic system (AI-FM) that enables the uninterrupted recognition and quantification of key mitophagic intermediates by extracting mitochondrial pH and morphological features. Using AI-FM, we identify a potential mitophagy modulator, Y040-7904, which enhances mitophagy by promoting mitochondria transport to autophagosomes and the fusion of autophagosomes with autolysosomes. Y040-7904 also reduces amyloid-β pathologies in both in vitro and in vivo models of Alzheimer's disease. This work offers an approach for visualizing the entire mitophagy flux, advancing the understanding of mitophagy-related mechanisms and enabling the discovery of mitophagy inducers for neurodegenerative diseases.

Authors

  • Yicheng Wang
    Shengli Clinical Medical College of Fujian Medical University, Fujian Medical University, Fuzhou, Fujian, China.
  • Pengfei Song
  • Heqing Zhou
    School of Pharmacy; MOE Key Laboratory of Smart Drug Delivery; MOE Innovative Center for New Drug Development of Immune Inflammatory Diseases; Zhongshan Hospital, Fudan University, Shanghai, China.
  • Pengwei Wang
    School of Information Science and Engineering, Shandong University, Qingdao, China. Electronic address: wangpw@sdu.edu.cn.
  • Yan Li
    Interdisciplinary Research Center for Biology and Chemistry, Liaoning Normal University, Dalian, China.
  • Zhiyong Shao
    State Key Laboratory of Medical Neurobiology and MOE Frontiers Center for Brain Science, Fudan University, Shanghai, China.
  • Lu Wang
    Department of Laboratory, Akesu Center of Disease Control and Prevention, Akesu, China.
  • Yan You
    Department of Pharmacology, School of Pharmacy, Fudan University, Shanghai, China. yyou@fudan.edu.cn.
  • Zuhai Lei
    Key Laboratory of Medicinal Chemistry for Natural Resource, Ministry of Education; School of Pharmacy, Yunnan University, Kunming, China. lei_zuhai@fudan.edu.cn.
  • Jinhua Yu
    Department of Electronic Engineering, Fudan University, Shanghai, 200433, China. jhyu@fudan.edu.cn.
  • Cong Li
    Key Laboratory of Synthetic and Natural Functional Molecule Chemistry of Ministry of Education, College of Chemistry and Materials Science, National Demonstration Center for Experimental Chemistry Education, Northwest University, Xi'an, Shaanxi 710127, China. Electronic address: licong@nwu.edu.cn.