AIMC Topic: Drug Discovery

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A comprehensive update on the application of high-throughput fluorescence imaging for novel drug discovery.

Expert opinion on drug discovery
INTRODUCTION: High-throughput fluorescence imaging (HTFI) is revolutionizing drug discovery by enabling rapid and precise detection of biological targets and cellular processes. Recent advances in fluorescence imaging technologies now provide unprece...

Natural language processing in drug discovery: bridging the gap between text and therapeutics with artificial intelligence.

Expert opinion on drug discovery
INTRODUCTION: The field of Natural Language Processing (NLP) within the life sciences has exploded in its capacity to aid the extraction and analysis of data from scientific texts in recent years through the advancement of Artificial Intelligence (AI...

TriCvT-DTI: Predicting Drug-Target Interactions Using Trimodal Representations and Convolutional Vision Transformers.

IEEE journal of biomedical and health informatics
Predicting interactions between drugs and their targets is vital for drug discovery and repositioning. Conventional techniques are slow and labor-intensive, while deep learning algorithms offer efficient solutions. However, deep learning often focus ...

DeepDTAGen: a multitask deep learning framework for drug-target affinity prediction and target-aware drugs generation.

Nature communications
Identifying novel drugs that can interact with target proteins is a highly challenging, time-consuming, and costly task in drug discovery and development. Numerous machine learning-based models have recently been utilized to accelerate the drug disco...

Advancements in Ligand-Based Virtual Screening through the Synergistic Integration of Graph Neural Networks and Expert-Crafted Descriptors.

Journal of chemical information and modeling
The fusion of traditional chemical descriptors with graph neural networks (GNNs) offers a compelling strategy for enhancing ligand-based virtual screening methodologies. A comprehensive evaluation revealed that the benefits derived from this integrat...

Artificial Intelligence in Molecular Optimization: Current Paradigms and Future Frontiers.

International journal of molecular sciences
Molecular optimization plays a pivotal role in many domains since it holds promise for improving the properties of lead molecules. The advent of artificial intelligence (AI)-driven molecular optimization has revolutionized lead optimization workflows...

Dumpling GNN: Hybrid GNN Enables Better ADC Payload Activity Prediction Based on the Chemical Structure.

International journal of molecular sciences
Antibody-drug conjugates (ADCs) are promising cancer therapeutics, but optimizing their cytotoxic payloads remains challenging. We present DumplingGNN, a novel hybrid Graph Neural Network architecture for predicting ADC payload activity and toxicity....

Machine Learning for Toxicity Prediction Using Chemical Structures: Pillars for Success in the Real World.

Chemical research in toxicology
Machine learning (ML) is increasingly valuable for predicting molecular properties and toxicity in drug discovery. However, toxicity-related end points have always been challenging to evaluate experimentally with respect to translation due to the re...

EnGCI: enhancing GPCR-compound interaction prediction via large molecular models and KAN network.

BMC biology
BACKGROUND: Identifying GPCR-compound interactions (GCI) plays a significant role in drug discovery and chemogenomics. Machine learning, particularly deep learning, has become increasingly influential in this domain. Large molecular models, due to th...

An AI-driven strategy for active compounds discovery and non-destructive quality control in traditional Chinese medicine: A case of Xuefu Zhuyu Oral Liquid.

Talanta
The modernization and globalization of traditional Chinese medicine (TCM) face challenges such as unclear active compounds and inadequate quality control. Taking Xuefu Zhuyu Oral Liquid (XZOL) as an example, this study proposed an artificial intellig...