AIMC Topic: Drug Discovery

Clear Filters Showing 1521 to 1530 of 1689 articles

An efficient curriculum learning-based strategy for molecular graph learning.

Briefings in bioinformatics
Computational methods have been widely applied to resolve various core issues in drug discovery, such as molecular property prediction. In recent years, a data-driven computational method-deep learning had achieved a number of impressive successes in...

DeepREAL: a deep learning powered multi-scale modeling framework for predicting out-of-distribution ligand-induced GPCR activity.

Bioinformatics (Oxford, England)
MOTIVATION: Drug discovery has witnessed intensive exploration of predictive modeling of drug-target physical interactions over two decades. However, a critical knowledge gap needs to be filled for correlating drug-target interactions with clinical o...

Pre-training graph neural networks for link prediction in biomedical networks.

Bioinformatics (Oxford, England)
MOTIVATION: Graphs or networks are widely utilized to model the interactions between different entities (e.g. proteins, drugs, etc.) for biomedical applications. Predicting potential interactions/links in biomedical networks is important for understa...

BACPI: a bi-directional attention neural network for compound-protein interaction and binding affinity prediction.

Bioinformatics (Oxford, England)
MOTIVATION: The identification of compound-protein interactions (CPIs) is an essential step in the process of drug discovery. The experimental determination of CPIs is known for a large amount of funds and time it consumes. Computational model has th...

Identifying drug-target interactions via heterogeneous graph attention networks combined with cross-modal similarities.

Briefings in bioinformatics
Accurate identification of drug-target interactions (DTIs) plays a crucial role in drug discovery. Compared with traditional experimental methods that are labor-intensive and time-consuming, computational methods are more and more popular in recent y...

Accelerating the discovery of antifungal peptides using deep temporal convolutional networks.

Briefings in bioinformatics
The application of machine intelligence in biological sciences has led to the development of several automated tools, thus enabling rapid drug discovery. Adding to this development is the ongoing COVID-19 pandemic, due to which researchers working in...

Big data and artificial intelligence (AI) methodologies for computer-aided drug design (CADD).

Biochemical Society transactions
There have been numerous advances in the development of computational and statistical methods and applications of big data and artificial intelligence (AI) techniques for computer-aided drug design (CADD). Drug design is a costly and laborious proces...

DD-GUI: a graphical user interface for deep learning-accelerated virtual screening of large chemical libraries (Deep Docking).

Bioinformatics (Oxford, England)
SUMMARY: Deep learning (DL) can significantly accelerate virtual screening of ultra-large chemical libraries, enabling the evaluation of billions of compounds at a fraction of the computational cost and time required by conventional docking. Here, we...

Artificial intelligence in the prediction of protein-ligand interactions: recent advances and future directions.

Briefings in bioinformatics
New drug production, from target identification to marketing approval, takes over 12 years and can cost around $2.6 billion. Furthermore, the COVID-19 pandemic has unveiled the urgent need for more powerful computational methods for drug discovery. H...