AIMC Topic: Quantitative Structure-Activity Relationship

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Machine Learning Modeling for ABC Transporter Efflux and Inhibition: Data Curation, Model Development, and New Compound Interaction Predictions.

Molecular pharmaceutics
In recent years, multiple computational studies have used machine learning models to predict substrate binding and inhibition of ATP-binding cassette (ABC) transporters. However, many of these studies relied on relatively small training sets with lim...

TRIumph in nanotoxicology: simplifying transcriptomics into a single predictive variable.

Nanoscale horizons
The primary aim of our study was to address the problem of transcriptomic data complexity by introducing a novel transcriptomic response index (TRI), compressing the entire transcriptomic space into a single variable, and linking it with the inhaled ...

Identification of novel DYRK1A inhibitors as treatment options for alzheimer's disease through comprehensive in silico approaches.

Scientific reports
This study aims to identify potential DYRK1A inhibitors from a curated database and utilize a QSAR model to predict the bioactivity of drug compounds in inhibiting the enzyme involved in tau protein oligomerization, a key process in AD pathology. 192...

Developing a predictive QSAR model for FGFR-1 inhibitors: integrating computational and experimental validation.

Journal of computer-aided molecular design
The traditional drug discovery process is often lengthy, costly, and characterized by a high failure rate. There is a pressing need for innovative strategies to optimize this process and improve the chances of identifying effective therapeutic candid...

Mathematical models for predicting the toxicity of micropollutant mixtures in water.

Arhiv za higijenu rada i toksikologiju
Water pollution caused by micropollutants has been a global issue for decades, prompting the scientific community and industry professionals to develop new and effective wastewater treatment methods. Understanding the interactions of these compounds ...

Design, Synthesis, and Aphicidal Activity of Novel Insect Neuropeptide Kinin Receptor Antagonists, Targeting the Ser Ligand Position.

Journal of agricultural and food chemistry
Traditional chemical pesticides have raised significant environmental and health concerns, driving the pursuit of safer alternatives. Aphids, notorious for causing extensive agricultural damage and transmitting plant diseases, represent prime targets...

Unveiling chemical space, scaffold diversity, critical structural features of pesticides: A comprehensive QSAR, qRASAR, machine learning studies to predict pesticides toxicity.

The Science of the total environment
The increasing use of pesticides in agriculture and urban areas has led to significant contamination of aquatic ecosystems, posing risks to non-target species. Fish, particularly the rainbow trout (Oncorhynchus mykiss), are highly vulnerable due to t...

From NMR to AI: Fusing H and C Representations for Enhanced QSPR Modeling.

Journal of chemical information and modeling
The ability to predict log  directly from spectral patterns marks a conceptual shift in cheminformatics. In this work, we demonstrate that H and C NMR spectra, computationally generated from molecular structures and transformed into machine learning-...

Frontiers Shaping the Next Generation of Transformation Product Prediction and Toxicological Assessment.

Environmental science & technology
The characterization of transformation products (TPs) is crucial for understanding chemical fate and potential environmental hazards. TPs form through (a)biotic processes and can be detected in environmental concentrations comparable to or even excee...

Predicting bone cancer drugs properties through topological indices and machine learning.

Scientific reports
Chemical graph theory and topological indices are key tools in the study of molecular structures and their properties. This research explores anticancer drugs using neighborhood degree-based topological indices and compares their efficacy through reg...