AIMC Topic: Drug Discovery

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DMAMP: A Deep-Learning Model for Detecting Antimicrobial Peptides and Their Multi-Activities.

IEEE/ACM transactions on computational biology and bioinformatics
Due to the broad-spectrum and high-efficiency antibacterial activity, antimicrobial peptides (AMPs) and their functions have been studied in the field of drug discovery. Using biological experiments to detect the AMPs and corresponding activities req...

Diffusing on Two Levels and Optimizing for Multiple Properties: A Novel Approach to Generating Molecules With Desirable Properties.

IEEE/ACM transactions on computational biology and bioinformatics
In the past decade, Artificial Intelligence (AI) driven drug design and discovery has been a hot research topic in the AI area, where an important branch is molecule generation by generative models, from GAN-based models and VAE-based models to the l...

An explainable deep learning platform for molecular discovery.

Nature protocols
Deep learning approaches have been increasingly applied to the discovery of novel chemical compounds. These predictive approaches can accurately model compounds and increase true discovery rates, but they are typically black box in nature and do not ...

Transforming drug discovery: the impact of AI and molecular simulation on R&D efficiency.

Bioanalysis
The process of developing new drugs in the pharmaceutical industry is both time-consuming and costly, making efficiency crucial. Recent advances in hardware and computational methods have led to the widespread application of computational science app...

Implementing enclosed sterile integrated robotic platforms to improve cell-based screening for drug discovery.

SLAS technology
At GSK, we have implemented custom integrated robotics platforms housed in bespoke biosafety enclosures to augment our capabilities in advanced cellular screening. Here we present and discuss the impact of one such system, the Cellular Automated Scre...

Self-Supervised Pre-Training via Multi-View Graph Information Bottleneck for Molecular Property Prediction.

IEEE journal of biomedical and health informatics
Molecular representation learning has remarkably accelerated the development of drug analysis and discovery. It implements machine learning methods to encode molecule embeddings for diverse downstream drug-related tasks. Due to the scarcity of labele...

Accelerating virtual patient generation with a Bayesian optimization and machine learning surrogate model.

CPT: pharmacometrics & systems pharmacology
The pharmaceutical industry has increasingly adopted model-informed drug discovery and development (MID3) to enhance productivity in drug discovery and development. Quantitative systems pharmacology (QSP), which integrates drug action mechanisms and ...

The Role of Artificial Intelligence and Machine Learning in Accelerating the Discovery and Development of Nanomedicine.

Pharmaceutical research
The unique potential of nanomedicine to address challenging health issues is rapidly advancing the field, leading to the generation of more effective products. However, these complex systems often pose several challenges with respect to their design ...

Structure-Aware Graph Attention Diffusion Network for Protein-Ligand Binding Affinity Prediction.

IEEE transactions on neural networks and learning systems
Accurate prediction of protein-ligand binding affinities can significantly advance the development of drug discovery. Several graph neural network (GNN)-based methods learn representations of protein-ligand complexes via modeling intermolecule intera...

A versatile attention-based neural network for chemical perturbation analysis and its potential to aid surgical treatment: an experimental study.

International journal of surgery (London, England)
Deep learning models have emerged as rapid, accurate, and effective approaches for clinical decisions. Through a combination of drug screening and deep learning models, drugs that may benefit patients before and after surgery can be discovered to red...