AI Medical Compendium Journal:
Journal of controlled release : official journal of the Controlled Release Society

Showing 1 to 10 of 21 articles

Integrity of polymeric micelles regulates bioavailability of cyclosporine A: A FRET-based analysis during oral delivery.

Journal of controlled release : official journal of the Controlled Release Society
This study comprehensively investigated the effect of structural integrity on the oral delivery efficacy of mPEG-b-PCL polymeric micelles (PMs) using fluorescence resonance energy transfer (FRET) technology. During mucus penetration, the integrity lo...

Dual-action membrane-chimeric liposomes with self-reinforcing targeting for acute lung injury treatment.

Journal of controlled release : official journal of the Controlled Release Society
Acute lung injury (ALI) is a common acute and critical syndrome with high mortality. The uncontrollable feedback loop of inflammation is the primary cause of death in patients with ALI. Therefore, targeting the inflammatory site and breaking the infl...

Dendritic cell-based microrobots for enhanced systemic antigen-specific immune tolerance.

Journal of controlled release : official journal of the Controlled Release Society
Current immunotherapeutic approaches for autoimmune disorders primarily rely on the use of generalized immunosuppressive medications. However, most immune drugs and tolerogenic immunomodulators are insufficient on their own to establish antigen-speci...

Active learning and Gaussian processes for the development of dissolution models: An AI-based data-efficient approach.

Journal of controlled release : official journal of the Controlled Release Society
In vitro dissolution testing plays a key role in controlling the quality and optimizing the formulation of solid dosage pharmaceutical products. Data-driven dissolution models can improve the efficiency of testing: their predictions can act as surrog...

AI-directed formulation strategy design initiates rational drug development.

Journal of controlled release : official journal of the Controlled Release Society
Rational drug development would be impossible without selecting the appropriate formulation route. However, pharmaceutical scientists often rely on limited personal experiences to perform trial-and-error tests on diverse formulation strategies. Such ...

Leveraging machine learning to streamline the development of liposomal drug delivery systems.

Journal of controlled release : official journal of the Controlled Release Society
Drug delivery systems efficiently and safely administer therapeutic agents to specific body sites. Liposomes, spherical vesicles made of phospholipid bilayers, have become a powerful tool in this field, especially with the rise of microfluidic manufa...

Optimizing lipid nanoparticles for fetal gene delivery in vitro, ex vivo, and aided with machine learning.

Journal of controlled release : official journal of the Controlled Release Society
There is a clinical need to develop lipid nanoparticles (LNPs) to deliver congenital therapies to the fetus during pregnancy. The aim of these therapies is to restore normal fetal development and prevent irreversible conditions after birth. As a firs...

Predicting tissue distribution and tumor delivery of nanoparticles in mice using machine learning models.

Journal of controlled release : official journal of the Controlled Release Society
Nanoparticles (NPs) can be designed for targeted delivery in cancer nanomedicine, but the challenge is a low delivery efficiency (DE) to the tumor site. Understanding the impact of NPs' physicochemical properties on target tissue distribution and tum...

Machine learning of Raman spectra predicts drug release from polysaccharide coatings for targeted colonic delivery.

Journal of controlled release : official journal of the Controlled Release Society
Colonic drug delivery offers numerous pharmaceutical opportunities, including direct access to local therapeutic targets and drug bioavailability benefits arising from the colonic epithelium's reduced abundance of cytochrome P450 enzymes and particul...

Machine learning in drug delivery.

Journal of controlled release : official journal of the Controlled Release Society
For decades, drug delivery scientists have been performing trial-and-error experimentation to manually sample parameter spaces and optimize release profiles through rational design. To enable this approach, scientists spend much of their career learn...